TAS-103 (dihydrochloride)

CAS No. 174634-09-4

TAS-103 (dihydrochloride) ( BMS-247615 dihydrochloride )

Catalog No. M20657 CAS No. 174634-09-4

TAS-103 (dihydrochloride) is a novel anticancer agent targeting both topoisomerase (Topo) I and Topo II.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 80 In Stock
10MG 120 In Stock
25MG 259 In Stock
50MG 385 In Stock
100MG 575 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    TAS-103 (dihydrochloride)
  • Note
    Research use only not for human use.
  • Brief Description
    TAS-103 (dihydrochloride) is a novel anticancer agent targeting both topoisomerase (Topo) I and Topo II.
  • Description
    TAS-103 (dihydrochloride) is a novel anticancer agent targeting both topoisomerase (Topo) I and Topo II.
  • Synonyms
    BMS-247615 dihydrochloride
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Topoisomerase
  • Recptor
    topo I/II
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    174634-09-4
  • Formula Weight
    406.31
  • Molecular Formula
    C20H21Cl2N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    H2O:50 mg/mL (123.06 mM; Need ultrasonic)
  • SMILES
    Cl.Cl.CN(C)CCNc1nc2cc(O)ccc2c2-c3ccccc3C(=O)c12
  • Chemical Name
    .6-((2-(dimethylamino)ethyl)amino)-3-hydroxy-7H-indeno[21-c]quinolin-7-one dihydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Aoyagi Y Kobunai T Utsugi T et al. In vitro Antitumor Activity of TAS-103 a Novel Quinoline Derivative That Targets Topoisomerases I and II[J]. Japanese journal of cancer research: Gann 1999 90(5):578-587.
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